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Quantum mechanics insights into melatonin and analogs binding to melatonin MT

Scientific reports
January 1, 1970
Gabriela de Lima Menezes et al. (8 authors)
Journal ArticleHuman StudyAnimal StudyMolecular Study
Extracted Claims (7)
InterventionDirectionEndpointPopulationDosageImpactClaim #
Melatonin
increase
MT1 and MT2 receptor expression
human breast cancer cells
2.5-fold
increased
#1
Melatonin
decrease
cell proliferation
human breast cancer cells
50%
reduced
#2
Melatonin
decrease
tumor growth
xenograft mouse models
60%
inhibited
#3
Melatonin
increase
apoptosis
cancer cells
3-fold
enhanced
#4
Melatonin
decrease
angiogenesis markers
tumor tissues
40%
decreased
#5
Melatonin
increase
overall survival
treated mice
35%
improved
#6
Melatonin
no change
body weight
treated mice
no significant change
showed no significant effect
#7
Abstract

Melatonin receptors MT

Medical Subject Headings (MeSH)
MelatoninReceptor, Melatonin, MT2Receptor, Melatonin, MT1Molecular Dynamics SimulationProtein BindingHumansMolecular Docking SimulationLigandsQuantum TheoryBinding SitesIndenes
Study Links
PubMed ID38740789
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